GPR75重组蛋白抗体
G蛋白偶联受体75(GPR75)为G蛋白偶联受体(GPCR)家族中的一员,是由 Tarttelin等人1999年首次发现,在肥胖、癌症和代谢综合征等许多疾病中发挥重要作用,是目前热手可热的减肥靶点之一。
GPR75之所以成为新兴的肥胖治疗靶点还是基于2021年7月Regeneron(再生元)在Science期刊上发表的研究。该研究通过对来自英国、美国和墨西哥的64.5万人的全外显子测序,分析罕见基因突变与体重指数(BMI)相关性,鉴定出16个非同义基因突变与BMI相关。其中,研究人员发现截短GPR75突变发生率为万分之四,杂合子突变BMI低1.8kg/㎡,体重轻5.4kg,肥胖概率低54%。该项研究中的小鼠体内验证试验表明,敲除GPR75小鼠体重更轻,血糖更低,胰岛素水平更低。更多关于GPR75靶点及信号通路>>
缔码生物科技有限公司是一家专注于可成药靶点临床前研发产品和服务的生物技术公司。缔码现可提供GPR75靶点全系列产品与服务。产品包括全长活性蛋白、ECD活性蛋白和流式验证单克隆抗体;服务包括多种属蛋白抗体定制服务、抗体人源化和亲和力成熟服务。此外,为加速GPR75生物疗法的开发,缔码还制备了GPR75靶点单B细胞种子库,最快28天可获得先导抗体分子。
ECD Proteins
SKU: PME-C100091 Target: GPR75
Price: 10μg ¥668.00 ; 50μg ¥2499.00 ; 100μg ¥3750.00
Overexpression Stable Cell Line
SKU: CEL100110 Target: GPR75
Application: FACS Data
Price: Inquiry
Overexpression Stable Cell Line
SKU: CEL100109 Target: GPR75
Application: FACS Data
Price: Inquiry
Full Length Transmembrane Proteins
SKU: FLP100031C Target: GPR75
Price: 10 μg ¥6300.00 ; 50 μg ¥30000.00 ; 100 μg ¥55000.00
Overexpression Stable Cell Line
SKU: CEL100092 Target: GPR75
Application: FACS Data
Price: Inquiry
Monoclonal Antibodies
PE-conjugated Anti-GPR75 antibody(DMC368); IgG1 Chimeric mAb
SKU: DMC100368P Target: GPR75
Application: Flow Cyt
Price: 100 test ¥3880.00
Monoclonal Antibodies
SKU: DME101136B Target: GPR75
Application: Flow Cyt
Price: 10μg ¥1030.00 ; 50μg ¥3380.00 ; 100 μg ¥6080.00 ; 500 μg ¥19880.00
Monoclonal Antibodies
SKU: DME101136 Target: GPR75
Application: Flow Cyt
Price: 10μg ¥690.00 ; 50μg ¥2280.00 ; 100 μg ¥4080.00 ; 500 μg ¥13280.00
Full Length Transmembrane Proteins
Human β2AR-GPR75-BRIL full length protein-synthetic nanodisc
SKU: FLP100031A Target: GPR75
Price: 10 μg ¥6300.00 ; 50 μg ¥30000.00 ; 100 μg ¥55000.00
Full Length Transmembrane Proteins
SKU: FLP110031 Target: GPR75
Price: 10 μg ¥6300.00 ; 50 μg ¥30000.00 ; 100 μg ¥55000.00
Full Length Transmembrane Proteins
SKU: FLP120031 Target: GPR75
Price: 10 μg ¥5670.00 ;50 μg ¥27000.00 ; 100 μg ¥49500.00
Monoclonal Antibodies
SKU: DMC100492B Target: GPR75
Application: Flow Cyt
Price: 10μg ¥1030.00 ; 50μg ¥3380.00 ; 100 μg ¥6080.00 ; 500 μg ¥19880.00
Monoclonal Antibodies
SKU: DMC100368B Target: GPR75
Application: Flow Cyt
Price: 10μg ¥1030.00 ; 50μg ¥3380.00 ; 100 μg ¥6080.00 ; 500 μg ¥19880.00
Monoclonal Antibodies
SKU: DMC100492 Target: GPR75
Application: Flow Cyt
Price: 10μg ¥690.00 ; 50μg ¥2280.00 ; 100 μg ¥4080.00 ; 500 μg ¥13280.00
ECD Proteins
SKU: PME101277 Target: GPR75
Price: 10μg ¥600.00 ; 50μg ¥2199.00 ; 100μg ¥3299.00
Full Length Transmembrane Proteins
SKU: FLP100031 Target: GPR75
Price: 10 μg ¥6300.00 ;50 μg ¥30000.00 ; 100 μg ¥55000.00
Monoclonal Antibodies
SKU: DMC100368 Target: GPR75
Application: Flow Cyt
Price: 10μg ¥690.00 ; 50μg ¥2280.00 ; 100 μg ¥4080.00 ; 500 μg ¥13280.00
ECD Proteins
SKU: PME100704 Target: GPR75
Price: 10μg ¥668.00 ; 50μg ¥2499.00 ; 100μg ¥3750.00
Monoclonal Antibodies
PE-conjugated Anti-GPR75 antibody(DMC492); IgG1 Chimeric mAb
SKU: DMC100492P Target: GPR75
Application: Flow Cyt
Price: 100 test ¥3880.00